Yohimbine HCL by MTS Nutrition | Kiss Those Trouble Areas GOODBYE!
What is Yohimbine HCl?
A lot of this information was learned from IFPA Pro Tommy Jeffers who was mentored by Lyle McDonald.
Yohimbe is harvested from trees grown in Africa and is used and sold as a supplement for fat loss and male sexuality. Yohimbine is a component of yohimbe and is the main alkaloid (and main active component) within yohimbe that produces the desired effects such as fat loss and male function (more shakin’ and bakin’).
We want the Yohimbine HCl—the ACTIVE EXTRACT-- not yohimbe bark which tends to not be accurately dosed. Thus, DO NOT BUY the bark, get the HCl version, as we make at MTS Nutrition. That way, we know what dose we are getting and can control the amount carefully, thus minimizing any side effects and maximizing results.
How Does Yohimbine HCl Work?
Yohimbine works on the alpha receptors. Alpha receptors inhibit fat breakdown, so wherever they are abundant, you have a harder time losing fat in that area. For example, they are in high concentration in men’s lower back and abs and in women’s hips and thighs. Yohimbine HCl acts as an alpha receptor blocker. Since alpha receptors inhibit fat breakdown, and Yohimbine HCl inhibits alpha receptors, the net result is that you get an INCREASE in fat breakdown. Thus, you get a significant increase in fat breakdown directly from an area that normally is the hardest place to lose it from. This is one reason why trainers like myself ALWAYS have my clients use this precontest!
Yohimbine HCL Dosage
Based on the studies we have examined, I recommend working up to 0.2mg/Kg of bodyweight. So that means a 220lb bodybuilder (divide by 2.2 to get Kg) is 100Kg and would work up to a dose of 20mg of Yohimbine HCl, or eight capsules of MTS Nutrition Yohimbine HCl. I would typically start this person at one capsule and work up towards the full dose each consecutive session the person had no undesirable side effects.
As I was discussing with Joe Daniels of Swing This Kettlebells, Yohimbine HCl's effects work the best in the absence of insulin, and its effects start to diminish the more insulin is present. But this doesn’t mean that you cannot eat carbs! Insulin will usually be under control on a lower carb diet, like most trainers will put you on. Obviously, cardio first thing in the morning is a good time (with a scoop of MTS Nutrition Whey in your belly) and even post workout. What you can do is take the Yohimbine HCl DURING your weight training workout 15-20 minutes before you are done. Then, hop on the cardio post weights and BAM—FAT BLAST!
Exclusively at TigerFitness.com!
Some studies on YHCl we used to extrapolate this data:1) Starke K, Trendelenburg AU, Limberger N. Presynaptic a 2-adrenoceptors: subtype determination. In: "Adrenoceptors: Structure, Function, and Pharmacology", Ruffolo, RR ed. Harwood Academic Publishers. 1995:99-108.
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3) Heible JP, Ruffolo RR, Starke K. Identification, characterization and subclassification of a 2-adrenoceptors: an overview. In: "a 2-Adrenergic Receptors: Structure, Function and Therapeutic Implications". Lanier SM, Limbird LE eds. Harwood Academic Press. 1997:1-18.
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6) Trendelenburg AU, Limberger N, Rump LC. a 2-Adrenergic receptors of the a 2C subtype mediate inhibition of norepinephrine release in human kidney cortex. Mol Pharmacol 1994; 415:M68-M76.
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49) Murburg MM, Villacres EC, Ko BN, Veith RC. Effects of yohimbine on human sympathetic nervous system function. J Clin Endocrin Metab 1991; 73:861-865.
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51) Henninger GR, Charney DS, Price LH. a 2-Adrenergic receptor sensitivity in depression. The plasma MHPG, behavioral and cardiovascular responses to yohimbine. Arc Gen Psychiatry 1988; 45:718-726.
52) McDougle CJ, Krystal JH, Price LH, Heninger GR, et al. Noradrenergic response to acute ethanol administration in healthy subjects: comparisons with intravenous yohimbine. Psychopharmacol 1995; 118:127-135.
53) Betz, JM, White KD. Gas chromatographic determination of yohimbine in commercial yohimbine products. J AOAC Int. 1995; 78:1189-1194.
54) Benedek IH, Blouin RA, McNamara PJ. Serum protein binding and the role of increased alpha1-acid glycoprotein in moderately obese subjects. Br J Clin Pharmacol 1984; 18:941-946.
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MTS Nutrition Yohimbine HCL 90 caps
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